T3 Liothyronine Sodium CAS 55-06-1 Oral anabolic steroid pauka no ka momona momona
Hōʻikeʻike wikiwiki
inoa huahana: Liothyronine Sodium (T3)
Alias: Cytomel T3;3, 3', 5-triiodothyronine sodium;T3
Einecs No: 200-223-5
MF: C15H11I3NNaO4
No CAS: 55-06-1
MW: 672.96
Maʻemaʻe: 99.0%
Nānā: keʻokeʻo i ka pauka beige
Hoʻohana: Hoʻoponopono pū kēia mau hormones i ka protein, ka momona, a me ka metabolism carbohydrate, e pili ana i ka hoʻohana ʻana o nā cell kanaka i nā pūhui ikaika.
T3 ka hoʻohana
Hana wikiwiki ʻo T3 i ka nalowale momona.Ma ke ʻano he alakaʻi, no ka hapa nui o 12.5 mcg/lā he ʻano "hoʻohui" conservative o ka dosing me he mea lā ʻaʻohe hopena ʻino i ka hana thyroid.
ʻO 25 mcg / lā he ʻano "hoʻohui" o ka dosing i loaʻa kekahi hopena pale.
ʻO 50 mcg / lā kahi ʻano bb'ing conservative kūpono, ʻoiaʻiʻo, ʻoi aku ka inhib.itori.
75 mcg / lā ke komo nei i loko o kahi wahi pilikia;
ʻO 100 mcg / lā i nā manawa he nui e alakaʻi i ka nalowale o ka nui a me ka ikaika.
Ma kēia ala, ʻo Liothyronine sodium, ʻo ka pahuhopu ka hoʻokō ʻana i kahi kihi mau i ka nalowale o ka momona a i ʻole ke kōkua.
e mālama i kahi hoʻonohonoho kino kokoke i ke kino.Ma kēia ala, haʻahaʻa loa ka dosing T3,
ʻoi aku ka maikaʻi o 12.5 mcg / lā akā i kekahi mau manawa e like me 25 mcg / lā.Ma ka ʻaoʻao haʻahaʻa o kēia pae, ʻaʻole e hōʻike ʻia ka hoʻāʻo thyroid ʻaʻole hiki ke ʻike ʻia me ka hoʻohana lōʻihi.Ma ka hopena kiʻekiʻe, ʻike ʻia ka hoʻopaʻa haʻahaʻa i kekahi manawa, akā ʻoi aku ka maikaʻi o nā hopena ma mua o ka lawe ʻole ʻia ʻana o T3, a hoʻohuli koke ka hoʻopau ʻana i ka hoʻopau ʻana i ka hoʻohana ʻana iā T3.
Ma ke ala ʻē aʻe, ʻo Liothyronine sodium, ʻo ka pahuhopu ke hoʻokō i kahi piʻi nui o ka momona o ka momona, ma ke kumukūʻai ʻike ʻia o ka hoʻoulu ʻana i ka hoʻopau ʻana i ka thyroid.ʻOi aku ka maikaʻi ma kahi o 50 mcg / lā, akā i kekahi mau manawa hiki ke kiʻekiʻe me 75 mcg / lā.ʻOi aku ka maikaʻi ʻaʻole e hoʻomau ʻia ka hoʻohana ʻana, akā no ka manawa palena wale e like me 8-12 pule, ʻoiai ʻaʻohe koi pololei no ka manawa.
T3 VS T4
Hoʻopau ʻia ʻo T4 e nā enzyme deiodinase ʻekolu e hana i ka triiodothyronine.
ʻO ka enzyme Deiodinase hoʻokahi ka helu no 80% o ka deiodination o T4, aia i loko o ke akepaʻa, ka puʻupaʻa, thyroid, a (i ka liʻiliʻi liʻiliʻi) pituitary.
Deiodinase enzyme 'elua makana i loko o CNS, pituitary, mediates manaʻo maikaʻi 'ole e pili ana i ka thyroid-stimulating hormone, a hāʻawi pū i loko o brown adipose kiko, a me ka puʻuwai moku, i ka predominantly intracellular.
ʻO ka enzyme Deiodinase ʻekolu, hoʻololi i ka T4 i T3 hoʻohuli, ʻaʻole like me T3, ʻaʻole hana, aia ia i loko o ka placenta, CNS, a me ka hemangioma.
T3 COA
Ka nana aku | He pauda ʻala ʻole, aneane keʻokeʻo a ʻulaʻula paha | hala |
Solubility | 1, hikiwawe loa i ka wai | hala |
2, hiki ke hoʻoheheʻe ʻia i ka waiʻona | hala | |
3, ʻaʻole hiki ke hoʻoheheʻe ʻia i ka hapa nui o nā mea hoʻoheheʻe organik | hala | |
4, hoʻoheheʻe ʻia i loko o ka wai hoʻoheheʻe sodium hydroxide | Holo | |
ʻIkepili | a) E wela ma kahi o 50 mg me nā kulu liʻiliʻi o ka ʻakika sulfuric i loko o kahi kīʻaha porcelain: ua hoʻomohala ʻia nā mahu waiola o ka iodine. | hala |
b) Hoʻopaʻa ʻia ka manawa paʻa o ka piko nui i ka RS | hala | |
Nalo ma ka maloo | ʻAʻole ʻoi aku ma mua o 4.0% | 0.46% |
[a]20/DC=1 in 1M HCl/EtOH 1:4 | +18 ~ +22o | +20.9o |
Hōʻike (HPLC) | ʻAʻole emi ma lalo o 95.0% | 99.18% |
ʻO ka sodium Levothyroxine | ʻAʻole ʻoi aku ma mua o 5.0% | 0.68% |
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